C102

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C102

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8-Cyclopentyl-1,3-dimethylxanthine

≥98% (HPLC), crystalline

Synonym:8-Cyclopentyltheophylline, CPT
CAS Number:35873-49-5
Linear Formula:C12H16N4O2
Molecular Weight:248.28
MDL number:MFCD00055116
PubChem Substance ID:24277730

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Description

Biochem/physiol ActionsSelective A1 adenosine receptor antagonist.

Properties

assay≥98% (HPLC)
formcrystalline
color white to off-white
solubilityH2O: <0.28 mg/mL, slightly soluble
 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.77 mg/mL
 DMSO: ~16 mg/mL at 60 °C
 0.1 M NaOH: soluble
Gene Informationhuman ... ADORA1(134)

Safety

Personal Protective EquipmentEyeshields, Gloves, type N95 (US), type P1 (EN143) respirator filter
WGK Germany3
RTECSXH5093600

References

referenceBruns, Adenosine antagonism by purines, pteridines and benzopteridines in human fibroblasts. Biochem. Pharmacol. 30, 325, (1981) Abstract
 Bruns, et al., Characterization of the A2 adenosine receptor labeled by [3H]NECA in rat striatal membranes. Mol. Pharmacol. 29, 331, (1986) Abstract